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Updated: Jun 22, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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血清素受体的阿洛斯特基调节剂:一种药物化学调查

Leonardo Brunetti1, Fabio Francavilla1, Marcello Leopoldo1

  • 1Department of Pharmacy-Drug Sciences, University of Bari Aldo Moro, 70125 Bari, Italy.

Pharmaceuticals (Basel, Switzerland)
|June 27, 2024
PubMed
概括

本综述探讨了血清素受体的全联体,重点是5-HT2C受体的天然化合物和合成调节剂. 这些全调节剂为诸如肥胖等疾病提供了传统药物潜在的更安全的替代品.

关键词:
在GPCR中,GPCR是指GPCR.基调节器是全基调节器.大麻素是一种大麻素.自然化合物 自然化合物血清胺 (serotonin) 是一种神经元.

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