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扎斯塔普拉赞的体外代谢和运输特征

Min Seo Lee1, Jihoon Lee2, Minyoung Pang3

  • 1College of Pharmacy and BK21 Four-Sponsored Advanced Program for SmartPharma Leaders, The Catholic University of Korea, Bucheon 14662, Republic of Korea.

Pharmaceutics
|June 27, 2024
PubMed
概括

扎斯塔普拉桑 (JP-1366) 是由药物代谢酶,主要是CYP3A4 / 3A5广泛代谢,影响其药理动力学. 药物运输体对斯塔普拉桑的吸收,分发和分泌的影响很小.

关键词:
毒品运输商 毒品运输商药物代谢酶的药物代谢酶.代谢物识别 代谢物识别具有竞争力的酸阻断剂 (P-CAB)斯塔普拉赞 (JP-1366) 是一个城市.

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