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Updated: Jun 22, 2025

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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通过氧化氨基化Cyclopentenones的Pyridones的合成简化

Bence B Botlik1, Micha Weber1, Florian Ruepp1

  • 1Laboratorium für Organische Chemie, ETH Zürich, Vladimir Prelog Weg 3, HCI, 8093, Zürich, Switzerland.

Angewandte Chemie (International ed. in English)
|June 27, 2024
PubMed
概括

研究人员开发了一种新的一方法,利用氧化氨基化来从环素中合成. 这种快速且可扩展的过程提供了一条简化通往有价值的胺化合物及其衍生物的途径.

关键词:
氨基化的氨基化.循环氨酸 (Cyclopentenones) 是一种含有循环氨酸的成分.过高价值的.皮里多尼酸盐 (pyridones) 是一种酸盐.环扩张 环扩张 环扩张

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