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Updated: Jun 22, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

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可光开关的美达博特罗普谷氨酸受体4的阳性全调节剂,以提高选择性

Silvia Panarello1,2, Aleix González-Díez1,2, Alice E Berizzi3

  • 1MCS, Institute for Advanced Chemistry of Catalonia - CSIC, Barcelona, Spain.

iScience
|July 5, 2024
PubMed
概括

研究人员开发了optogluram-2,一种新型的可光开关联体,用于甲基胺基质受体4 (mGlu4). 这种化合物提供了增强的选择性和精确的光控制调制,有助于神经系统疾病研究.

关键词:
生物化学 生物化学生物科学 生物科学分子生物学分子生物学自然科学自然科学自然科学药理学 药理学 药理学 药理学 药理学

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