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Updated: Jun 21, 2025

Quantifying Agonist Activity at G Protein-coupled Receptors
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M2肌糖受体对抗剂和全调节剂的电压依赖性

Shimrit Hazan1, Merav Tauber1, Yair Ben-Chaim1

  • 1Department of Natural Sciences, The Open University of Israel, Ra'anana, Israel.

Biochemical pharmacology
|July 12, 2024
PubMed
概括

研究了肌肉蛋白受体对抗剂的电压依赖性. 阿特罗平和斯科波胺显示了电压依赖的功效,而AF-DX 386则没有,为GPCR药理学提供了新的见解.

关键词:
其他模块化模块.敌对者的敌对者G 蛋白结合受体的受体.肌肉性受体是指肌肉性受体.电压依赖性 电压依赖性在Xenopus的卵细胞中.

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