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Updated: Jun 20, 2025

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

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选择性地将插入到基中

Zheng Zhang1, Qi Li1, Zengrui Cheng2

  • 1Department of Chemistry, Institute of Molecular Plus, Tianjin Key Laboratory of Molecular Optoelectronic Science, School of Pharmaceutical Science and Technology, Tianjin University, Tianjin, China.

Nature communications
|July 17, 2024
PubMed
概括

这项研究引入了一种新的分子编辑策略,用于合成含化合物. 该方法有效地将插入基中,使得能够创建有价值的制药中间体和药物修饰.

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