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Updated: Jun 20, 2025

Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding
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能驱动G蛋白结合受体亚型中的联体识别

Xin Yang1,2, Pei Zhou1,2, Siyuan Shen1

  • 1Department of Biotherapy, State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, Chengdu, Sichuan 610041, China.

Proceedings of the National Academy of Sciences of the United States of America
|July 18, 2024
PubMed
概括

研究人员发现了大麻素受体 (CB) 亚型选择性的驱动机制. 这一发现使得能够合理设计具有高度选择性的药物,具有较低的成潜力.

关键词:
在GPCR中,GPCR是指GPCR.发现药物的发现.进入的过程中,连接器识别 连接器识别分子动力学模拟模拟

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