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Updated: Jun 20, 2025

A High-throughput Calcium-flux Assay to Study NMDA-receptors with Sensitivity to Glycine/D-serine and Glutamate
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作为神经元离子通道阻断剂的N-硫烯素

Matthieu Schmit1,2, Md Mahadhi Hasan3, Yashad Dongol3

  • 1School of Chemistry, Monash University Victoria 3800 Australia Kellie.Tuck@monash.edu.

RSC medicinal chemistry
|July 19, 2024
PubMed
概括

新的N-sulfonylphenoxazines通过有效抑制N型通道来治疗神经性疼痛具有前景. 这些化合物表现出更好的稳定性和潜在的血脑屏障透,提供了新的治疗途径.

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