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Updated: Jun 18, 2025

Rapid In Situ Hybridization using Oligonucleotide Probes on Paraformaldehyde-prefixed Brain of Rats with Serotonin Syndrome
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释放高分子量5-HT7R配体的潜力:合成,亲和力和ADMET检查

Patryk Pyka1, Sabrina Garbo2, Aleksandra Murzyn3

  • 1Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University, Medical College, Medyczna 9, PL 30-688 Kraków, Poland; Doctoral School of Medical and Health Sciences, Jagiellonian University Medical College, 31-530 Kraków, Poland.

Bioorganic chemistry
|July 30, 2024
PubMed
概括

研究人员开发了针对中枢神经系统疾病的5-HT7受体的新型aryl-piperazine hydantoin配体. 一种化合物显示出有前途的类似药物的特性和治疗神经退行性疾病的潜力.

关键词:
在ADMET中,ADMET的属性是:停靠对接 停靠对接与G蛋白结合的受体是G蛋白结合的受体.基因表达测试试验在MTS测试中,测量分子建模分子建模血清素受体5-HT ((7)) 的使用.在体外实验实验

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