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Updated: Jun 18, 2025

Simultaneous Measurement of HDAC1 and HDAC6 Activity in HeLa Cells Using UHPLC-MS
09:20

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Published on: August 10, 2017

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针对癌症治疗HDAC6的小分子:目前的进展和新的策略

Ziqian Huang1, Ling Li2, Binbin Cheng3

  • 1Department of Pharmacy, First Affiliated Hospital of Gannan Medical University, Ganzhou 341000, PR China.

Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie
|July 31, 2024
PubMed
概括

基因组脱乙酶6 (HDAC6) 是一种关键的癌症标. 像双作用抑制剂和向蛋白降解 (TPD) 这样的新策略显示出在癌症治疗中克服传统HDAC6抑制剂的局限性的希望.

关键词:
生物功能的生物功能.双目标抑制剂 双目标抑制剂希斯脱乙酶6 (HDAC6) 是一种选择性抑制剂 选择性抑制剂有针对性的蛋白质降解 (TPD)

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