通过 (-) - 大麻烯激活CB2受体,但不通过 (+) - 大麻烯激活CB2受体

Michael Udoh1, Marina Santiago1, Syed Haneef1

  • 1Macquarie Medical School, Macquarie University, North Ryde, Australia.

PubMed
概括

该研究发现, (-) - 卡纳比克罗 (CBC) 是CB2受体中的活性反体,而 (-) - 卡纳比克罗和 (+) - 卡纳比克罗都激活TRPA1通道. 药用CBC制剂可能更有效,具有主导 (-) -CBC.

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