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Updated: Jun 15, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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普罗托帕纳克萨迪醇衍生物:一种具有抗炎作用的新型选择性葡萄皮质受体调节剂的植物原产物

Zhenyuan Li1, Teng Liu1, Wenbin Xie1

  • 1School of Pharmacy, Key Laboratory of Molecular Pharmacology and Drug Evaluation (Yantai University), Ministry of Education, Collaborative Innovation Center of Advanced Drug Delivery System and Biotech Drugs in Universities of Shandong, Yantai University, Yantai, 264005, Shandong, PR China.

European journal of pharmacology
|August 24, 2024
PubMed
概括

一种植物化合物SP-8像选择性葡萄皮质受体调节器 (SGRM) 一样起作用. 它通过抑制NF-κB通路而减少炎症,而不会引起典型的葡萄糖皮质体副作用,为炎症性疾病治疗提供了潜力.

关键词:
这是一种抗炎症的药物.葡萄糖皮质类受体受体这是一种Proto-panaxadiol.选择性葡萄糖皮质体受体调节器交易激活 交易激活转压抑是一种转压抑.

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