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Updated: Jun 15, 2025

Modification and Functionalization of the Guanidine Group by Tailor-made Precursors
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2H-P2Y6受体对手的功能化原生

Paola Oliva1, Asmita Pramanik1, Young-Hwan Jung1

  • 1Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, MD 20892, USA.

Cells
|August 28, 2024
PubMed
概括

具有长链氨基酸修饰的新型P2Y6受体对抗剂显著增强了亲和力和选择性. 这些化合物,特别是类似物30 (MRS4940),显示出治疗炎症和退行性疾病的潜力.

关键词:
在GPCR中,GPCR是指GPCR.这是一个P2Y受体.作为一个对抗者的对抗者.和是最重要的.核酸核酸是一种核酸.结构活动关系结构活动关系

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