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Updated: Jun 14, 2025

Facile Preparation of 4-Substituted Quinazoline Derivatives
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Published on: February 15, 2016

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作为高效的A2A腺素受体对抗剂的新奇基纳佐林衍生物

Amélie Laversin1, Robin Dufossez1, Raphaël Bolteau1

  • 1Univ. Lille, Inserm, CHU Lille, U1172-LilNCog-Lille Neuroscience & Cognition, F-59000 Lille, France.

Molecules (Basel, Switzerland)
|August 29, 2024
PubMed
概括

研究人员开发了新型的2-aminoquinazoline衍生物作为腺A2A受体 (A2AR) 对抗剂. 这些化合物显示出治疗神经退行性疾病和癌症的前景,通过增强目标亲和力和可溶性.

关键词:
它是A2A受体对抗剂.这是一种cAMP测试.光的两极化是因为光.氨酸氨酸是一种氨酸.

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