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Updated: Jun 14, 2025

In Vitro Imaging and Quantification of the Drug Targeting Efficiency of Fluorescently Labeled GnRH Analogues
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Published on: March 21, 2017

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确定针对生长激素释放激素受体 (GHRHR) 的小分子对手

Minos-Timotheos Matsoukas1, Tarryn Radomsky2,3, Vasilis Panagiotopoulos1

  • 1University of West Attica, Department of Biomedical Engineering, Athens 12243, Greece.

Journal of chemical information and modeling
|August 29, 2024
PubMed
概括

研究人员确定了生长激素释放激素受体 (GHRHR) 的第一个非类对抗剂,这是癌症治疗的有前途标. 这些新型的小分子在体外显示出抑制GHRH活性的潜力.

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