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Updated: Jun 14, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Published on: February 20, 2018

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GPR56/ADGRG1的G蛋白选择性概况及其对下游效应器的影响

Raida Jallouli1,2, Ana L Moreno-Salinas1,2, Andréanne Laniel1,2

  • 1Department of Pharmacology-Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, Québec, Canada.

Cellular and molecular life sciences : CMLS
|September 4, 2024
PubMed
概括

不同的GPR56配体通过不同的机制激活受体,影响G蛋白选择性. 这些通路汇聚在Rho通路激活上,这对于GPR56在生理和癌症环境中的功能至关重要.

关键词:
布雷特·布雷特是什么意思G蛋白结合受体的受体是G蛋白结合受体的受体.在 GPR56 中使用.罗格埃夫 (RhoGEF) 是一个类型.信号传输 信号传输人口贩运 人口贩运

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