新的皮里米丁衍生物与西林对抗抗甲素耐药的金黄色葡萄球菌的协同效应

Bruna Kelly de Oliveira Silva1, Zenaide Severina do Monte1, Erick Caique Santos Costa2

  • 1Postgraduate Program in Pharmaceutical Sciences-Federal University of Pernambuco, Av. Prof. Moraes Rego, 1235 - University City, Recife, PE, 50740-560, Brazil.

Future medicinal chemistry
|September 5, 2024
PubMed
概括

一种新型的pyrimidine化合物,PYB01,通过调节Staphylococcus aureus的耐药性机制,显示出对抗抗菌素耐药性的潜力. 这种化合物表现出适度的抗生素活性和有利的药理动力学特性.