FL118:,H2A.X,

Guangrui Fan1, Xiongfei Luo2, Yibo Shi1

  • 1Institute of Urology, Lanzhou University Second Hospital, Urinary System Disease Clinical Medical Research Center of Gansu Province, NO. 82 Cuiying Gate, Lanzhou 730000, Gansu Province, China.

Bioorganic chemistry
|September 8, 2024
PubMed
概括

一种新型化合物FL118通过抑制细胞增殖和克服凝素+青抗性,有效向膀癌. 它充当分子,结合H2A.X和DNA,诱导细胞亡并阻碍DNA修复.