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Updated: Jun 13, 2025

Optimizing the Genetic Incorporation of Chemical Probes into GPCRs for Photo-crosslinking Mapping and Bioorthogonal Chemistry in Live Mammalian Cells
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Optimizing the Genetic Incorporation of Chemical Probes into GPCRs for Photo-crosslinking Mapping and Bioorthogonal Chemistry in Live Mammalian Cells

Published on: April 9, 2018

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为PGC1α招募调RXR调节器

Felix Nawa1, Minh Sai1, Jan Vietor1

  • 1Department of Pharmacy, Ludwig-Maximilians-Universität (LMU) München, 81377 Munich, Germany.

Journal of medicinal chemistry
|September 11, 2024
PubMed
概括

合成激动剂选择性地将PGC1α招募到核视网体X受体 (RXRs),与内源性配体不同. 这种选择性核心调节器调节为基于RXR的向治疗提供了潜力.

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