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Updated: Jun 13, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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多组分帕塞里尼反应作为一种方法来获得结构,活性和性质的多样性:软硬的化物/大麻素调节器

Angela Lamberti1, Marta Serafini2, Silvio Aprile2

  • 1Instituto de Investigación, Desarrollo e Innovación en Biotecnología Sanitaria de Elche (IDiBE), Universidad Miguel Hernández, Elche, Spain.

European journal of medicinal chemistry
|September 12, 2024
PubMed
概括

研究人员探索了内分泌体 (EV) /内分泌体 (EC) 系统,发现了针对炎症和疼痛的新化合物. 化合物41作为TRPV1和CB2受体的平衡激动剂具有良好的代谢稳定性.

关键词:
这些受体是CB CB受体.双重定位是双重的目标.帕塞里尼的多元件反应反应多种药理学 多种药理学软毒品是一种软毒品.在 TRPV1 频道.

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