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Updated: Jun 13, 2025

Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors
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基于循环butan的小分子αvβ3抗剂的侧链结构-活性关系

Adam Throup1, Manar Saleh Zraikat1, Andrew Gordon1

  • 1Institute of Cancer Therapeutics, University of Bradford Bradford BD7 1DP UK h.sheldrake@bradford.ac.uk.

RSC medicinal chemistry
|September 16, 2024
PubMed
概括

研究人员使用功能化循环butanes开发了新的整合素抗剂. 这种有前途的方法针对癌症和其他疾病,其中一种化合物显示出良好的体外和体内结果,以便进一步开发.

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