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Updated: Jun 13, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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GPR56/ADGRG1的G蛋白选择性概况及其对下游效应器的影响

Raida Jallouli1, Ana Lilia Moreno Salinas1, Andréanne Laniel1

  • 1Université de Sherbrooke: Universite de Sherbrooke.

Research square
|September 16, 2024
PubMed
概括

不同的GPR56配体通过不同的机制激活受体,影响癌细胞中的G蛋白选择性和Rho通路激活. 这一发现为研究GPR56活性及其在癌症中的作用提供了新的工具.

关键词:
布雷特·布雷特是什么意思G蛋白结合受体的受体是G蛋白结合受体的受体.在 GPR56 中使用.罗格埃夫 (RhoGEF) 是一个类型.信号传输 信号传输走私和贩运的人口贩运

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