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Updated: Jun 12, 2025

Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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乳糖酶介导的5-aminopyrazoles的化学选择性C-4化

Mansour Shahedi1, Rojina Shahani1, Niloofar Omidi1

  • 1Department of Organic Chemistry, Shahid Beheshti University, Tehran, Iran.

PloS one
|September 18, 2024
PubMed
概括

研究人员开发了一种使用laccase酶对5-aminopyrazoles进行化学选择性 arylation的新方法. 这种高效的工艺避免了恶劣的条件,并产生了有价值的C-4化化合物.

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