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Updated: Jun 12, 2025

A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors
10:28

A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors

Published on: August 17, 2019

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人类F-ATP合成酶作为药物标

Christoph Gerle1, Chimari Jiko2, Atsuki Nakano3

  • 1Life Science Research Infrastructure Group, RIKEN SPring-8 Center, Kouto, 1-1-1, Sayo, Hyogo, Japan.

Pharmacological research
|September 20, 2024
PubMed
概括

人类F-ATP合成酶对细胞能量至关重要,具有治疗潜力. 本综述探讨了其功能,并确定了开发新药治疗人类疾病的结构性目标.

关键词:
这是ATP合成酶.的 FoF1 ATP 酶.奥克斯福斯 (OXPHOS) 是一个药物设计 药物设计膜蛋白质是一种膜蛋白质.线粒体中的线粒体.

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