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Updated: Jun 12, 2025

A Semi-Quantitative Drug Affinity Responsive Target Stability DARTS assay for studying Rapamycin/mTOR interaction
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Published on: August 27, 2019

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拉帕米辛抑制剂的目标哺乳动物水平在博治疗下降

Lena-Luise Becker1, Karen Agricola2, David M Ritter2

  • 1Institute of Cell Biology and Neurobiology, Department of Pediatric Neurology, Center for Chronically Sick Children, Charité-Universitätsmedizin Berlin, Berlin, Germany.

Pediatric neurology
|September 21, 2024
PubMed
概括

在瘤硬化综合体 (TSC) 患者中,使用乳腺胺抑制剂 (mTORi) 向哺乳动物的塞诺巴马特导致埃弗罗利斯水平显著下降. 建议监测mTORi水平,当与cenobamate同时使用时.

关键词:
基酸盐 (Cenobamate) 是一种这是Everolimus.这就是西罗利木斯.结核性硬化综合体 结核性硬化综合体这是一种mTOR抑制剂.

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