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Updated: Jun 10, 2025

Functionalized Spirocyclic Heterocycle Synthesis and Cytotoxicity Assay
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以多样性为导向的战略 (DOS) 用于高效合成具有抗癌活性的福[2,3-b]二衍生物

Reymark Ereje1,2, Jantana Yahuafai3, Theeranuch Jaroenchuensiri1

  • 1Center of Excellence in Natural Products, Department of Chemistry, Faculty of Science, Chulalongkorn University, Pathumwan, Bangkok, 10330, Thailand.

ChemMedChem
|October 18, 2024
PubMed
概括

通过以多样性为导向的合成 (DOS) 合成了新的硫胺 (BFP) 衍生物. 一些类型显示强大的抗癌活性和对癌细胞的选择性,提供有前途的治疗线索.

关键词:
本佐福罗皮里丁 (benzofuropyridine) 是一种天然的酸盐.癌症 癌症 癌症 癌症药物发现 药物发现分子对接是分子对接.在QSAR分析中,分析了QSAR.

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