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Updated: Jun 9, 2025

Autoradiography as a Simple and Powerful Method for Visualization and Characterization of Pharmacological Targets
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Published on: March 12, 2019

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结构-亲和力-药物动力学关系的新 18 F-标记的1,4-亚泽衍生物的奥雷克辛1受体成像

Yui Ishizaka1, Hiroyuki Watanabe1, Masahiro Ono1

  • 1Department of Patho-Functional Bioanalysis, Graduate School of Pharmaceutical Sciences, Kyoto University, 46-29 Yoshida Shimoadachi-cho, Sakyo-ku, Kyoto 606-8501, Japan.

Journal of medicinal chemistry
|October 21, 2024
PubMed
概括

研究人员开发了一种新的放射性追踪剂[18F]BTF,用于使用正子发射断层扫描 (PET) 绘制素1受体 (OX1R) 的图像. 这种追踪器对可视化大脑中的OX1R和推进药物开发具有前途.

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