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Updated: Jun 9, 2025

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皮拉佐利胺 - 基合物:合成和抗基因菌体活性

Devesh S Agarwal1, Richard M Beteck1, Dorien Mabille2

  • 1Centre of Excellence for Pharmaceutical Sciences, North-West University, Potchefstroom, 2520, South Africa.

Naunyn-Schmiedeberg's archives of pharmacology
|October 21, 2024
PubMed
概括

新的pyrazolyl amide-chalcones被合成并对kinetoplastid寄生虫进行了测试. 化合物9b对Trypanosoma brucei brucei具有很高的活性,而9n对Trypanosoma brucei rhodesiense具有很强的活性.

关键词:
氨基酸氨基化物 氨基酸氨基化物这是一种抗尼内托塑的药物.哈尔科内斯 (Chalcones) 是一种石头.药物相似性属性 药物相似性属性这些是Pyrazoles.

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