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探索具有抗癌作用的COX抑制剂的结构-活性关系:综合性综述

Ozlem Akgul1, Mustafa Gul2, Halise Inci Gul3

  • 1Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Ege University, 35100 Bornova, İzmir-Turkey.

Current topics in medicinal chemistry
|October 23, 2024
PubMed
概括

向循环氧化酶-2 (COX-2) 显示出癌症治疗的前景. 选择性COX-2抑制剂,特别是具有二异环基架的抑制剂,对癌细胞表现出显著的细胞毒性活性.

关键词:
抗氧化抑制剂 (COX抑制剂) 的使用在COX-2中,COX-2是最常见的.这是一种抗癌药物.这是一种抗炎药,抗炎药.药物开发是药物的发展.结构-活动关系关系.

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