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作为具有抗炎和抗氧化性质的选择性COX-2抑制剂的pyrimidine衍生物

Beata Tylińska1, Anna Janicka-Kłos2, Tomasz Gębarowski3

  • 1Department of Organic Chemistry, Wroclaw Medical University, Borowska 211A, 50-556 Wroclaw, Poland.

International journal of molecular sciences
|October 26, 2024
PubMed
概括

新的胺衍生物L1和L2通过选择性抑制循环氧化酶-2 (COX-2) 和减少炎症细胞生长,显示出强大的抗炎作用. 这些化合物还具有抗氧化特性,并与白蛋白结合,这表明开发更安全的药物的潜力.

关键词:
抑制COX的抑制作用癌症治疗疗法 癌症治疗这是一种炎症炎症炎症炎症.

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