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Updated: May 6, 2026

Systemic and Local Drug Delivery for Treating Diseases of the Central Nervous System in Rodent Models
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在老鼠中中枢神经系统和脑后神经系统中未结合的eletriptan和sumatriptan的区域分布:对潜在的中心作用的影响

Nana Svane1, Frida Bällgren2, Aghavni Ginosyan2

  • 1Department of Pharmacy, CNS Drug Delivery and Barrier Modelling group (CNSBM), University of Copenhagen, Copenhagen, Denmark.

The journal of headache and pain
|October 31, 2024
PubMed
概括

三药有效地治疗偏头痛,通过达到外周和中枢神经系统的受体. 尽管血脑屏障的透能力有限,但eletriptan和sumatriptan实现了显著的5-HT受体占用,这表明在偏头痛治疗中可能存在潜在的中心机制.

关键词:
5-HT1B / 1D / 1F受体的受体血液-大脑屏障是什么?在CNS中,CNS是CNS.中心效应是中心效应.组合绘图方法是一种组合绘图方法.埃利特里普坦是什么意思 埃利特里普坦免费药物理论是什么偏头痛是一种偏头痛.在PNS中,使用PNS.苏马特里普坦是苏马特里普坦的一个.

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