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Updated: Jun 8, 2025

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Published on: June 13, 2022

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新型二硫胺含有双二醇部分,具有选择性碳酸酶抑制和抗癌活性

Aida Buza1, Cüneyt Türkeş2, Mustafa Arslan3

  • 1Department of Chemistry, Faculty of Mathematical and Natural Sciences, University of Prishtina Prishtina 1000 Republic of Kosova arleta.rifati@uni-pr.edu.

RSC medicinal chemistry
|November 4, 2024
PubMed
概括

新的硫胺化合物被合成为人类碳酸酶 (hCA) 抑制剂. 几种化合物显示出对与瘤相关的hCA IX和XII的强大和选择性抑制,其中一些也显示出选择性癌细胞细胞毒性.

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