针对表皮生长因子受体 (EGFR) 的生理活性异环体混合的综合分析和结果

Mandeep Kaur1, Hafiz Muzzammel Rehman2, Yurong Wu3

  • 1Synthetic and Medicinal Chemistry Laboratory, Department of Chemistry, Punjabi University, Patiala, 147002, India.

PubMed
概括

这项研究开发了新型化合物来抑制癌症中的表皮生长因子受体 (EGFR). 化合物7和8通过有效向非活性和突变EGFR形式,显示出作为抗癌剂的显著潜力.

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