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Updated: Jun 7, 2025

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最近在开发17β-hydroxysteroid脱酶抑制剂方面取得的进展

Donald Poirier1

  • 1Laboratory of Medicinal Chemistry, Endocrinology and Nephrology Unit, CHU de Québec Research Center-Université Laval, Québec, QC G1V 4G2, Canada; Department of Molecular Medicine, Faculty of Medicine, Université Laval, Québec, QC G1V 0A6, Canada.

Steroids
|November 12, 2024
PubMed
概括

本综述强调了最近在开发17β-hydroxysteroid脱酶 (17β-HSDs) 选择性抑制剂方面取得的进展. 这些抑制剂向各种17β-HSD异型,为荷尔蒙依赖性疾病提供潜在的治疗策略.

关键词:
17β-HSDD 的使用情况.药物设计 药物设计酵素酶是一种酶.激素 激素是一种激素.抑制剂的抑制剂类固醇的产生.

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