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C2230,一种优先使用和状态依赖的CaV2.2通道阻断剂,可以在多种疼痛模型中减轻疼痛行为

Cheng Tang1,2,3, Kimberly Gomez4, Yan Chen3

  • 1Department of Molecular Pathobiology, College of Dentistry, and.

The Journal of clinical investigation
|December 10, 2024
PubMed
概括

一种新的CaV2.2抑制剂C2230通过选择性抑制N型通道,为慢性疼痛管理提供了一种新的方法. 这种化合物有望开发出更安全,更有效的止痛药,副作用更少.

关键词:
通道是一种通道.神经科学是一个神经科学.疼痛 疼痛 疼痛 疼痛药理学 药理学 是一个学科.

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