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Updated: Jun 5, 2025

Author Spotlight: Streamlining Protein Target Prediction and Validation via Molecular Docking and CETSA
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根据它们的向结合位点对共价蛋白结合剂进行分类

Walaa A Bedewy1, John W Mulawka2, Marc J Adler2

  • 1Department of Chemistry & Biology, Toronto Metropolitan University, Toronto, ON M5B 2K3, Canada; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Egypt.

Bioorganic & medicinal chemistry letters
|December 12, 2024
PubMed
概括

联蛋白结合剂现在被认为是安全和有效的治疗方法,提供诸如增强的功效和对突变的抵抗等优势. 本综述探讨了它们在药物发现中的多样化的结合部位和应用.

关键词:
同价药物药物是共价药物.蛋白质结合剂 蛋白质结合剂

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