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Updated: Jun 5, 2025

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药物设计的最新发展口服合成自由脂肪酸受体1激动剂

Lei Liu1,2, Qinghua Zhang1,2, Yichuan Ma3

  • 1Tasly Academy, Tasly Pharma Co., Ltd., Tianjin, People's Republic of China.

Drug design, development and therapy
|December 16, 2024
PubMed
概括

合成FFAR1激动剂在糖尿病和肝病方面表现有前途,但肝毒性仍然是一个挑战. 模仿天然产品的新型低分子量化合物提供了改善的肝脏安全性和潜在的治疗益处.

关键词:
抗糖尿病药物 抗糖尿病药物人工智能辅助的人工智能辅助人工智能基于脂肪酸的脂毒性肝毒性 肝毒性 肝毒性以自然为灵感的结构修改.口头 FFAR1 的发展.

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