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Updated: Jun 4, 2025

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine

Published on: June 13, 2022

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通过基质氨基转移方法对Sacubitril的立体选择性合成的研究

Megha V Sadanande1,2, Sagar S Thorat1,2, Himanshu Sharma2,3

  • 1Organic Chemistry Division, CSIR-National Chemical Laboratory, Dr. Homi Bhabha Road, Pune, 411008, India.

Chemistry, an Asian journal
|December 23, 2024
PubMed
概括

我们开发了新型合成路径,用于sacubitril,一个关键的 neprilysin 抑制剂. 这些方法利用奇拉氨基转移试剂进行高效的立体选择性合成,改善药物制造.

关键词:
基质氨基转移 (CAT) 方法.奇拉式池方法的方法.萨库比特里尔 (Sacubitril) 是一种药物.立体选择性合成

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