通过顺序的催化Aza-Heck/苏苏基合反应对Isoindolinone进行选择性合成

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Updated: Jun 4, 2025

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

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Lei Wang1, Wenyu Zhang1, Shuaijie Wu1

  • 1School of Chemistry & Chemical Engineering, Yangzhou University, Yangzhou, Jiangsu 225002, China.

Organic letters
|December 23, 2024
PubMed
概括

一个新的tandem aza-Heck/Suzuki交叉合反应有效地合成了奇拉性isoindolinones. 这种由催化的方法在温和条件下使用O-基乙烯和酸,实现高反选择性.

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