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Drug Delivery: Overview
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The selection of a drug's delivery route depends upon its physicochemical properties, including lipid or water solubility and ionization, as well as the therapeutic requirement, such as immediate or sustained effect. These routes can be divided into three primary categories: enteral, parenteral, and topical.
Enteral delivery involves administering drugs directly through swallowing, sublingual placement, or buccal application. Orally administered drugs predominantly navigate the...
Enteral delivery involves administering drugs directly through swallowing, sublingual placement, or buccal application. Orally administered drugs predominantly navigate the...
276
Drug Delivery: Miscellaneous Routes
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Drug delivery methods like oral inhalation, nasal sprays, transdermal patches, eye drops, intravitreal injection, and rectal administration provide localized effects with reduced toxicity.
Oral inhalation and nasal sprays swiftly transfer drugs across the respiratory epithelium's mucosal layer. Inhaled glucocorticoids and bronchodilators directly target lung conditions such as asthma, while fluticasone nasal spray mitigates allergic rhinitis.
Transdermal patches transport drugs...
Oral inhalation and nasal sprays swiftly transfer drugs across the respiratory epithelium's mucosal layer. Inhaled glucocorticoids and bronchodilators directly target lung conditions such as asthma, while fluticasone nasal spray mitigates allergic rhinitis.
Transdermal patches transport drugs...
315
Drug Delivery: Parenteral Route
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The parenteral route is a critical method of drug administration. It delivers compounds directly into the systemic circulation and bypasses the gastrointestinal tract. This approach is particularly advantageous for drugs that exhibit poor absorption or instability when administered orally.
There are three primary parenteral routes: intravenous (IV), intramuscular (IM), and subcutaneous (SC). The IV route introduces the drug directly into the bloodstream, ensuring immediate action. The IM route...
There are three primary parenteral routes: intravenous (IV), intramuscular (IM), and subcutaneous (SC). The IV route introduces the drug directly into the bloodstream, ensuring immediate action. The IM route...
411
Drug Delivery: Enteral Route
377
The enteral drug administration involves three primary routes: oral, sublingual, and buccal. Oral ingestion is the most prevalent, safe, economical, and convenient method for drug administration. However, it has certain drawbacks, including limited absorption due to the drug's low water solubility or poor membrane permeability, possible emesis from GI mucosa irritation, destruction of drugs by digestive enzymes or low gastric pH, and irregular absorption along with food or other drugs.
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Routes of Drug Administration: Parenteral
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The administration of drugs via parenteral routes allows for direct drug introduction into the systemic circulation, resulting in high bioavailability because the medication bypasses the harsh conditions of the gastrointestinal tract and hepatic metabolism.
The intravenous route (IV) of drug administration can be further categorized into two types. The bolus injection administers the entire dose rapidly, while an intravenous infusion slowly delivers smaller doses steadily.
The IV route is often...
The intravenous route (IV) of drug administration can be further categorized into two types. The bolus injection administers the entire dose rapidly, while an intravenous infusion slowly delivers smaller doses steadily.
The IV route is often...
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Mechanisms of Drug Absorption: Paracellular, Transcellular, and Vesicular Transport
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Drugs need to permeate cell membranes to reach their target sites after administration. Orally administered drugs must transcend intestinal epithelial membrane barriers to infiltrate the systemic circulation. Drugs with a molecular weight of less than 500 Daltons diffuse through gaps between neighboring cells, called paracellular pathways.
However, most drugs use the transcellular route, traversing directly through the cell membranes via two mechanisms: passive and active transport. Passive...
However, most drugs use the transcellular route, traversing directly through the cell membranes via two mechanisms: passive and active transport. Passive...
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基于离子二极管的药物输送系统
Hyunjae Yoo1, Soon-Bo Kang1, Jeongsoo Kim2
1Department of Material Science and Engineering, Seoul National University, Seoul, 08826, Republic of Korea.
Advanced materials (Deerfield Beach, Fla.)
|December 24, 2024
概括
一种新的离子二极管药物递送系统可以控制细胞毒药物的持续释放,提高抗瘤疗效,并在临床前模型中降低毒性.
科学领域:
- 生物医学工程 生物医学工程
- 材料科学 材料科学 材料科学
- 在瘤学瘤学.
背景情况:
- 传统的药物输送系统在与细胞毒性药物的空间时间控制和持续释放作斗争.
- 实现精确的药物释放对于最大限度地提高疗效和最大限度地减少非目标组织损伤至关重要.
研究的目的:
- 开发和评估一种基于电位控制的离子二极管的药物输送系统,用于持续和局部的药物释放.
- 在临床前瘤模型中评估该系统的抗瘤疗效和安全性.
主要方法:
- 一个离子二极管系统被设计用于通过电势控制药物释放 (纳米到微克尺度).
- 该系统使用水凝来缓慢,连续地将药物扩散到目标部位.
- 该装置植入了一个自由移动的携带瘤的小鼠模型中,并加载了多克索鲁比辛.
主要成果:
- 离子二极管系统证明了持续的,无流量药物输送,在长时间内泄漏最小.
- 在体内研究表明,与内注射相比,通过系统输送的多克索鲁比辛的抗瘤疗效优越.
- 该系统表现出最小的非目标免疫毒性,突出其安全性.
结论:
- 离子二极管药物递送系统为控制和持续释放细胞毒剂提供了一个有希望的平台.
- 该系统的生物兼容性和机械兼容性支持其在治疗手术无法切除的瘤方面的临床转化潜力.


