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Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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合成和抗微生物活性评价含有伊米达佐提亚迪亚佐尔部分的皮拉衍生物

Lan-Ying Han1, Jing-Xin Sun1, Chuang Liu1

  • 1Key Laboratory of Natural Medicines of the Changbai Mountain, Ministry of Education, College of Pharmacy, Yanbian University, Yanji, China.

Future medicinal chemistry
|December 26, 2024
PubMed
概括

新的皮拉衍生物对抗多药耐药菌株表现出强大的抗菌活性. 化合物23h具有高效和安全性,表明其作为一种新型抗菌剂的潜力.

关键词:
皮拉 (Pyrazole) 是一种可怕的药物.抗微生物活性的抗微生物活性.血液溶解 (hemolysis) 是一种imidazo[2,1-b][1,3,4]thiadiazole的使用情况多种药物耐药性多种药物耐药性

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