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Updated: Jun 3, 2025

A Semi-Quantitative Drug Affinity Responsive Target Stability DARTS assay for studying Rapamycin/mTOR interaction
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用天然化合物准mTOR激酶:通过增强的结合机制强大的ATP竞争性抑制

Sulaiman K Marafie1, Eman Alshawaf1, Fahd Al-Mulla2

  • 1Biochemistry and Molecular Biology Department, Dasman Diabetes Institute, Dasman 15462, Kuwait.

Pharmaceuticals (Basel, Switzerland)
|January 8, 2025
PubMed
概括

传统中医药中的两种天然化合物有效地抑制了拉巴胺素 (mTOR) 激酶域 (KD) 的哺乳动物标. 这些化合物表现出稳定的结合,为与mTOR失调相关的疾病提供潜在的新疗法.

关键词:
这就是ATPATPATPATP.激酶域域名 激酶域名在mTOROR中使用mTOR.这是一种mTOR抑制剂.分子模拟分子模拟自然化合物 自然化合物

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