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Updated: Jun 2, 2025

Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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基于分子对接的设计和开发的pyrazol-5-ylbenzamide衍生物含有奇拉性oxazoline部分作为杀菌剂

Xiang Cheng1, Zhen Zhang1, Yuanjian Huang1

  • 1College of Materials and Chemistry and School of Plant Protection, Anhui Agricultural University, Hefei, China.

Pest management science
|January 16, 2025
PubMed
概括

新型性pyrazol-5-yl-benzamide衍生物显示强大的抗真菌活性对抗Valsa mali. 这些化合物,特别是 (S) -4h,为作物保护提供了有希望的替代品,降低了耐药性风险,对蜜蜂没有毒性.

关键词:
急性口服毒性急性口服毒性这是一种性真菌杀菌剂.分子对接的分子对接.分子动力学模拟,分子动力学模拟这种药物是oxazoline.简化脱酶的作用.理论上的计算,理论上的计算.

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