MimoSamycin Janus 2 :

Kamonpan Sanachai1, Kowit Hengphasatporn2, Supakarn Chamni3

  • 1Center of Excellence in Structural and Computational Biology, Department of Biochemistry, Faculty of Science, Chulalongkorn University, Bangkok 10330, Thailand.

概括

咪索氨酸有效地抑制了Janus酶2 (JAK2),这是白血病发展中的关键蛋白质. 这项研究探讨了它的机制,并为潜在的白血病治疗设计了改进的抑制剂.