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Updated: May 31, 2025

High-throughput Screening for Small-molecule Modulators of Inward Rectifier Potassium Channels
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High-throughput Screening for Small-molecule Modulators of Inward Rectifier Potassium Channels

Published on: January 27, 2013

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针对的Kv7通道作为的目标

Emilio Perucca1,2, Maurizio Taglialatela3

  • 1Department of Medicine (Austin Health), Melbourne Brain Center, The University of Melbourne, 245 Burgundy St., Heidelberg, VIC, 3084, Australia. emilio.perucca@unimelb.edu.au.

CNS drugs
|January 24, 2025
PubMed
概括

电压关联的Kv7通道是治疗的关键目标. 新的Kv7.2/7.3激活剂,如阿泽图卡纳,在抗药性发作中显示出有前途,比较老药物提供了更好的安全性.

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