Dandan Sha1, Minghui Yuan1, Lin Zhang2

  • 1Jiangsu Collaborative Innovation Center of Biomedical Functional Materials, Jiangsu Key Laboratory of Biomedical Materials, School of Chemistry and Materials Science, Nanjing Normal University, Nanjing, 210023, China.

概括

胆酸,如陶罗胆酸 (TCA) 和糖胆酸 (GCA),与胰岛素非共价结合,增强口服生物可用性. 质谱学显示,TCA与胰岛素的结合力比GCA更强.