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为了增强生物活动和稳定性,对 Cordycepin 衍生物的分子工程

Yiming Gu1, Wei Yu1, Xiang Li2

  • 1State Key Laboratory of Metastable Materials Science and Technology, Nano-biotechnology Key Lab of Hebei Province, Applying Chemistry Key Lab of Hebei Province, Yanshan University, Qinhuangdao, 066004, China.

ChemMedChem
|February 5, 2025
PubMed
概括

新型cordycepin衍生物被合成,以克服由腺脱氨酶 (ADA) 引起的代谢不稳定性. 五种衍生品表现出增强的抗菌活性和改善的稳定性,提供了潜在的治疗进展.

关键词:
具有抗菌活性,具有抗菌活性.它具有抗瘤活性.在Cordycepin衍生品中.与ADA相比,稳定性是非常重要的.

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