相关实验视频

Updated: May 27, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

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设计,合成和GluN2A负基调节器的表征,适用于体外勘探

François P Bischoff1, Sven Van Brandt1, Marcel Viellevoye1

  • 1Janssen Research & Development, Janssen Pharmaceutica NV, Turnhoutseweg 30, B-2340 Beerse, Belgium.

Journal of medicinal chemistry
|February 17, 2025
PubMed
概括

研究人员开发了新的工具来研究GluN2A受体,这些受体对学习和记忆至关重要. 这些来自MPX-004和MPX-007的新型化合物显示出对N-甲基-D-酸盐受体体体内研究的改善特性.

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A High-throughput Calcium-flux Assay to Study NMDA-receptors with Sensitivity to Glycine/D-serine and Glutamate04:48

A High-throughput Calcium-flux Assay to Study NMDA-receptors with Sensitivity to Glycine/D-serine and Glutamate

Published on: July 10, 2018

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