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Updated: May 27, 2025

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发现了新型pH敏感的μ-阿片类受体激活剂,作为具有减少副作用的强效止痛药

Zhen Wang1,2, Zong-Zheng Li2, Xiao-Min Han2

  • 1School of Pharmaceutical Sciences, Hubei University of Medicine, Shiyan 442000, China.

ACS medicinal chemistry letters
|February 19, 2025
PubMed
概括

一种新型的pH敏感化合物,22,选择性地准片受体 (MOR) 来缓解疼痛. 这种新的止痛药证明了效果,副作用比传统阿片类药物少.

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