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Updated: May 27, 2025

Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding
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Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding

Published on: June 9, 2017

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通过多个Gαi/o异形,CB1受体与细胞外调节激酶的合

Boyd R Rorabaugh1,2, Daniel J Morgan1,2

  • 1Department of Pharmaceutical Sciences, Marshall University School of Pharmacy.

Neuroreport
|February 20, 2025
PubMed
概括

大麻素1型受体 (CB1Rs) 通过多个Gαi/o蛋白激活细胞外信号调节激酶 (ERK). 这项研究确定了Gαo,Gαi1,Gαi2和Gαi3作为合伙伴,Gαi3可能对部分激素激剂诱导的ERK激活至关重要.

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